Table 2

List of P-glycoprotein substrates

Substrate
Steroid compounds
    Aldosterone
    Progesterone
    Hydrocortisone
    Cortisol
    Corticosterone
    Dexamethasone
Anticancer agents
    Doxorubicin
    Daunorubicin
    Vinca alkaloids
    Actinomycin D
    Epotoside
Immunosuppressive agents
    Cyclosporin
    FK 506
    Methotrexate
Protease inhibitors
    Indinavir
    Nelfinavir
    Ritonavir
Antibiotics
    Erythromycin
    Rifampicin
Cardiac drugs
    Digoxin
    Quinidine
    Lovastatin
Antihistamines
    Terfenadine
Others
    Domperidone
    Loperamide